Morpholine catalyzed direct C3 alkenylation of indoles with α,β-unsaturated aldehydes.

نویسندگان

  • Shi-Kai Xiang
  • Bo Zhang
  • Li-He Zhang
  • Yuxin Cui
  • Ning Jiao
چکیده

Organocatalytic direct C3 alkenylation of indoles has been developed. Simple and readily available morpholine trifluoroacetic acid salt is employed as an efficient catalyst in this oxidative dehydrogenative reaction. Simplicity and practicality constitute the most attractive advantages of this reaction.

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عنوان ژورنال:
  • Chemical communications

دوره 47 28  شماره 

صفحات  -

تاریخ انتشار 2011